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A Metabolic Function for Phospholipid and Histone Methylation: Molecular Cell
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Other agonists, such as the intestine-specific Fexaramine D (FexD), suppressed colitis-associated cancer (CAC) by restoring FXR signaling, enhancing intestinal barrier integrity, and reducing pro-inflammatory M1-like macrophage infiltration within the TIME ( Conversely, FXR inhibition or functional antagonism demonstrates therapeutic value where FXR activation is detrimental